Identification of the GPR55 Agonist Binding Site Using a Novel Set of High-Potency GPR55 Selective Ligands-Reference-Cited by-同舟云学术

Identification of the GPR55 Agonist Binding Site Using a Novel Set of High-Potency GPR55 Selective Ligands

Published:2011-06-01 Issue:25 Volume:50 Page:5633-5647
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Kotsikorou Evangelia¹,Madrigal Karla E.¹,Hurst Dow P.¹,Sharir Haleli²,Lynch Diane L.¹,Heynen-Genel Susanne³,Milan Loribelle B.³,Chung Thomas D. Y.³,Seltzman Herbert H.⁴,Bai Yushi⁵,Caron Marc G.⁵,Barak Larry⁵,Abood Mary E.²,Reggio Patricia H.¹

Affiliation:

1. Center for Drug Discovery, University of North Carolina, Greensboro, North Carolina 27402, United States

2. Department of Anatomy and Cell Biology and Center for Substance Abuse Research, Temple University, Philadelphia, Pennsylvania 19140, United States

3. Conrad Prebys Center for Chemical Genomics at Sanford-Burnham Medical Research Institute, La Jolla, California 92037, United States

4. Center for Organic and Medicinal Chemistry, Research Triangle Institute, Research Triangle Park, North Carolina 27709, United States

5. Department of Cell Biology, Duke University, Durham, North Carolina 27708, United States

Publisher

American Chemical Society (ACS)

Subject

Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/bi200010k

Reference57 articles.

1. Identification and cloning of three novel human G protein-coupled receptor genes GPR52, ΨGPR53 and GPR55: GPR55 is extensively expressed in human brain

2. The putative cannabinoid receptor GPR55 plays a role in mechanical hyperalgesia associated with inflammatory and neuropathic pain

3. The putative cannabinoid receptor GPR55 affects osteoclast function in vitro and bone mass in vivo

4. A role for L-α-lysophosphatidylinositol and GPR55 in the modulation of migration, orientation and polarization of human breast cancer cells

5. The orphan G protein-coupled receptor GPR55 promotes cancer cell proliferation via ERK

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