Novel Oxadiazole Analogues Derived from Ethacrynic Acid: Design, Synthesis, and Structure−Activity Relationships in Inhibiting the Activity of Glutathione S-Transferase P1-1 and Cancer Cell Proliferation-Reference-Cited by-同舟云学术

Novel Oxadiazole Analogues Derived from Ethacrynic Acid: Design, Synthesis, and Structure−Activity Relationships in Inhibiting the Activity of Glutathione S-Transferase P1-1 and Cancer Cell Proliferation

Published:2010-01-07 Issue:3 Volume:53 Page:1015-1022
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Yang Xinmei¹,Liu Guyue²,Li Hongcai¹,Zhang Yun¹,Song Dandan²,Li Chunmin¹,Wang Rui³,Liu Bo¹,Liang Wen¹,Jing Yongkui³,Zhao Guisen¹

Affiliation:

1. School of Pharmaceutical Sciences, Shandong University, Jinan, Shandong 250012, P. R. China

2. Shenyang Pharmaceutical University, Shenyang 110016, P. R. China

3. Mount Sinai School of Medicine, One Gustave L. Levy Place, New York, New York 10029

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9011565

Reference30 articles.

1. The role of glutathione-S-transferase in anti-cancer drug resistance

2. Overexpression of glutathione S-transferase π enhances the adduct formation of cisplatin with glutathione in human cancer cells

3. Glutathione S—transferase and drug resistance

4. Glutathione-S-transferase π inhibits As2O3-induced apoptosis in lymphoma cells: involvement of hydrogen peroxide catabolism

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