Process Research and Development and Scale-up of a 4,4-Difluoro-3,3-dimethylproline Derivative-Reference-Cited by-同舟云学术

Process Research and Development and Scale-up of a 4,4-Difluoro-3,3-dimethylproline Derivative

Published:2008-02-21 Issue:2 Volume:12 Page:322-338
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Rossi Francesco¹,Corcella Francesco¹,Caldarelli Francesco Saverio¹,Heidempergher Franco¹,Marchionni Chiara¹,Auguadro Miriam¹,Cattaneo Marco¹,Ceriani Lucio¹,Visentin Giuseppina¹,Ventrella Giambattista¹,Pinciroli Vittorio¹,Ramella Giuliano¹,Candiani Ilaria¹,Bedeschi Angelo¹,Tomasi Attilio¹,Kline Billie J.¹,Martinez Carlos A.¹,Yazbeck Daniel¹,Kucera David J.¹

Affiliation:

1. Active Pharmaceutical Ingredients and Analytical Development & Quality Control, Nerviano Medical Sciences, Pharmaceutical Sciences Unit Viale Pasteur 10, 20014 Nerviano, Italy, and Chemical Research and Development, La Jolla Laboratories, Pfizer Inc., 10578 Science Center Drive, San Diego, California 92121-1111, U.S.A.

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op7001112

Reference28 articles.

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2. Kucera, D. J.; Saeed, N. L.; Scott, R. W.PCT Int. Appl. 2005054187, 2005.

3. Catalysis of the Cope and Claisen rearrangements

4. Claisen rearrangement of allyl esters

5. The ester enolate Claisen rearrangement. Stereochemical control through stereoselective enolate formation

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