ST7612AA1, a Thioacetate-ω(γ-lactam carboxamide) Derivative Selected from a Novel Generation of Oral HDAC Inhibitors-Reference-Cited by-同舟云学术

ST7612AA1, a Thioacetate-ω(γ-lactam carboxamide) Derivative Selected from a Novel Generation of Oral HDAC Inhibitors

Published:2014-10-08 Issue:20 Volume:57 Page:8358-8377
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Giannini Giuseppe¹,Vesci Loredana¹,Battistuzzi Gianfranco¹,Vignola Davide¹,Milazzo Ferdinando M.¹,Guglielmi Mario Berardino¹,Barbarino Marcella¹,Santaniello Mosè¹,Fantò Nicola¹,Mor Marco²,Rivara Silvia²,Pala Daniele²,Taddei Maurizio³,Pisano Claudio¹,Cabri Walter¹

Affiliation:

1. R&D Sigma-Tau Industrie Farmaceutiche Riunite SpA, Via Pontina Km 30,400, I-00040 Pomezia, Roma, Italy

2. Dipartimento di Farmacia, Università degli Studi di Parma, Parco Area delle Scienze 27/A, I-43124 Parma, Italy

3. Dipartimento di Biotecnologie, Chimica e Farmacia, Università degli Studi di Siena, Via A. Moro 2, I-53100 Siena, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm5008209

Reference59 articles.

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4. Endogenous modulators and pharmacological inhibitors of histone deacetylases in cancer therapy

5. Histone deacetylase inhibitors in the treatment of cancer: overview and perspectives

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