An Efficient, Stereoselective Synthesis of the Hydroxyethylene Dipeptide Isostere Core for the HIV Protease Inhibitor A-792611-Reference-Cited by-同舟云学术

An Efficient, Stereoselective Synthesis of the Hydroxyethylene Dipeptide Isostere Core for the HIV Protease Inhibitor A-792611

Published:2006-06-09 Issue:14 Volume:71 Page:5369-5372
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Engstrom Kenneth¹,Henry Rodger¹,Hollis L. Steven¹,Kotecki Brian¹,Marsden Ian¹,Pu Yu-Ming¹,Wagaw Seble¹,Wang Weifeng¹

Affiliation:

1. Department of Process Chemistry, Department of Structural Chemistry, Global Pharmaceutical Research and Development, Abbott Laboratories, 1401 Sheridan Road, North Chicago, Illinois 60064-6290 seble.wagaw@abbott.com

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo060737s

Reference10 articles.

1. Peptidomimetic Inhibitors of HIV Protease

2. Chiral synthetic intermediates via asymmetric hydrogenation of .alpha.-methyl-.alpha.,.beta.-unsaturated aldehydes by bakers' yeast

3. HIV-1 protease inhibitors based on hydroxyethylene dipeptide isosteres: An investigation into the role of the P1' side chain on structure-activity

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