Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5-HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers-Reference-Cited by-同舟云学术

Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5-HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers

Published:2012-11-09 Issue:22 Volume:55 Page:9693-9707
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Dubost Emmanuelle¹,Dumas Noé²,Fossey Christine¹,Magnelli Rosa¹,Butt-Gueulle Sabrina¹,Ballandonne Céline¹,Caignard Daniel H.³,Dulin Fabienne¹,Sopkova de-Oliveira Santos Jana¹,Millet Philippe²,Charnay Yves²,Rault Sylvain¹,Cailly Thomas¹,Fabis Frederic¹

Affiliation:

1. UFR des Sciences Pharmaceutiques, Université de Caen Basse-Normandie, EA 4258 CERMN, FR CNRS 3038 INC3M, SF-4206 ICORE, Boulevard Becquerel, F-14032 Caen, France

2. Unité de Morphologie et Unité de Neuroimagerie, Service de Neuropsychiatrie, Hôpitaux Universitaires de Genève, Ch. du Petit-Bel-Air, 2, CH1225 Chêne-Bourg/Genève, Switzerland

3. Institut de Recherches Servier, 125 Chemin de Ronde, F-78290 Croissy sur Seine, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300943r

Reference57 articles.

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2. Review of 5-HT4R Ligands: State of Art and Clinical Applications

3. Serotonin Receptors, Type 4: A New Hope?

4. Serotonin pharmacology in the gastrointestinal tract: a review

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