Reduction of Peptide Character of HIV Protease Inhibitors That Exhibit Nanomolar Potency against Multidrug Resistant HIV-1 Strains-Reference-Cited by-同舟云学术

Reduction of Peptide Character of HIV Protease Inhibitors That Exhibit Nanomolar Potency against Multidrug Resistant HIV-1 Strains

Published:2003-03-18 Issue:9 Volume:46 Page:1764-1768
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tamamura Hirokazu¹,Koh Yasuhiro¹,Ueda Satoshi¹,Sasaki Yoshikazu¹,Yamasaki Tomonori¹,Aoki Manabu¹,Maeda Kenji¹,Watai Yoriko¹,Arikuni Hisashi¹,Otaka Akira¹,Mitsuya Hiroaki¹,Fujii Nobutaka¹

Affiliation:

1. Graduate School of Pharmaceutical Sciences, Kyoto University, Sakyo-ku, Kyoto 606-8501, Japan; Department of Internal Medicine II, Kumamoto University School of Medicine, Kumamoto 860-8556, Japan; Yokohama Laboratory, SC BioSciences Corporation, Hodogaya-ku, Yokohama 240-0005, Japan; and Experimental Retrovirology Section, Medicine Branch, Division of Clinical Sciences, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020537i

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3. L-735,524: an orally bioavailable human immunodeficiency virus type 1 protease inhibitor.

4. ABT-538 is a potent inhibitor of human immunodeficiency virus protease and has high oral bioavailability in humans.

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