Nonpolar and Short Side Chain Groups at C-11β of Estradiol Result in Antiestrogens-Reference-Cited by-同舟云学术

Nonpolar and Short Side Chain Groups at C-11β of Estradiol Result in Antiestrogens

Published:2005-02-10 Issue:5 Volume:48 Page:1428-1447
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zhang Jing-xin¹,Labaree David C.¹,Hochberg Richard B.¹

Affiliation:

1. Department of Obstetrics/Gynecology and Reproductive Sciences, and the Comprehensive Cancer Center, Yale University School of Medicine, New Haven, Connecticut 06520

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049352x

Reference41 articles.

1. Estradiol-16α-carboxylic Acid Esters as Locally Active Estrogens

2. Synthesis and Evaluation of B-, C-, and D-Ring-Substituted Estradiol Carboxylic Acid Esters as Locally Active Estrogens

3. The estradiol pharmacophore: Ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site

4. A Simple and Sensitive Microtiter Plate Estrogen Bioassay Based on Stimulation of Alkaline Phosphatase in Ishikawa Cells: Estrogenic Action of Δ5Adrenal Steroids*

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