Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloid Receptor Antagonist-Reference-Cited by-同舟云学术

Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloid Receptor Antagonist

Published:2004-11-12 Issue:6 Volume:48 Page:1857-1872
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Swanson Devin M.¹,Dubin Adrienne E.¹,Shah Chandra¹,Nasser Nadia¹,Chang Leon¹,Dax Scott L.¹,Jetter Michele¹,Breitenbucher J. Guy¹,Liu Changlu¹,Mazur Curt¹,Lord Brian¹,Gonzales Lisa¹,Hoey Kenway¹,Rizzolio Michele¹,Bogenstaetter Michael¹,Codd Ellen E.¹,Lee Doo H.¹,Zhang Sui-Po¹,Chaplan Sandra R.¹,Carruthers Nicholas I.¹

Affiliation:

1. Johnson & Johnson Pharmaceutical Research and Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, and Johnson & Johnson Pharmaceutical Research and Development L.L.C., Welsh and McKean Roads, Spring House, Pennsylvannia 19477

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0495071

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