Skeletal Editing Approach to Bridge-Functionalized Bicyclo[1.1.1]pentanes from Azabicyclo[2.1.1]hexanes-Reference-Cited by-同舟云学术

Skeletal Editing Approach to Bridge-Functionalized Bicyclo[1.1.1]pentanes from Azabicyclo[2.1.1]hexanes

Published:2023-05-05 Issue:20 Volume:145 Page:10960-10966
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Wright Brandon A.¹^ORCID,Matviitsuk Anastassia²^ORCID,Black Michael J.¹,García-Reynaga Pablo²,Hanna Luke E.²,Herrmann Aaron T.²,Ameriks Michael K.²^ORCID,Sarpong Richmond¹^ORCID,Lebold Terry P.²

Affiliation:

1. Department of Chemistry, University of California, Berkeley, California 94720, United States

2. Janssen Research and Development, San Diego, California 92121, United States

Funder

Janssen Research and Development

Division of Graduate Education

University of California

National Institute of General Medical Sciences

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/jacs.3c02616

Reference63 articles.

1. The importance of synthetic chemistry in the pharmaceutical industry

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5. Application of the Bicyclo[1.1.1]pentane Motif as a Nonclassical Phenyl Ring Bioisostere in the Design of a Potent and Orally Active γ-Secretase Inhibitor

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