Tripeptide Aldehyde Inhibitors of Human Rhinovirus 3C Protease: Design, Synthesis, Biological Evaluation, and Cocrystal Structure Solution of P1 Glutamine Isosteric Replacements-Reference-Cited by-同舟云学术

Tripeptide Aldehyde Inhibitors of Human Rhinovirus 3C Protease: Design, Synthesis, Biological Evaluation, and Cocrystal Structure Solution of P1 Glutamine Isosteric Replacements

Published:1998-06-26 Issue:15 Volume:41 Page:2786-2805
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Webber Stephen E.¹,Okano Koji¹,Little Thomas L.¹,Reich Siegfried H.¹,Xin Yue¹,Fuhrman Shella A.¹,Matthews David A.¹,Love Robert A.¹,Hendrickson Thomas F.¹,Patick Amy K.¹,Meador James W.¹,Ferre Rose Ann¹,Brown Edward L.¹,Ford Clifford E.¹,Binford Susan L.¹,Worland Stephen T.¹

Affiliation:

1. Agouron Pharmaceuticals, Inc., 3565 General Atomics Court, San Diego, California 92121

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm980071x

Reference56 articles.

1. (a) Couch, R. B. Rhinoviruses. InVirology; Fields, B. N., Knipe, D. M., Eds.; Raven Press: New York, 1990; Volume 1, Chapter 22, pp 607−629.

2. TREATMENT OF THE PICORNA VIRUS COMMON COLD BY INHIBITORS OF VIRAL UNCOATING AND ATTACHMENT

3. RHINOVIRUS COLDS

4. (d) Gwaltney, J. M. Rhinoviruses. InViralInfections of Humans; Evans, A. S., Ed.; Plunem Publishing Corp. New York, 1982; Chapter 20, pp 491−517.

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