Design and Synthesis of Photoaffinity-Labeling Ligands of the l-Prolyl-l-leucylglycinamide Binding Site Involved in the Allosteric Modulation of the Dopamine Receptor-Reference-Cited by-同舟云学术

Design and Synthesis of Photoaffinity-Labeling Ligands of the l-Prolyl-l-leucylglycinamide Binding Site Involved in the Allosteric Modulation of the Dopamine Receptor

Published:2005-11-30 Issue:1 Volume:49 Page:307-317
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Fisher Abigail¹,Mann Amandeep¹,Verma Vaneeta¹,Thomas Nancy¹,Mishra Ram K.¹,Johnson Rodney L.¹

Affiliation:

1. Department of Medicinal Chemistry, University of Minnesota, 308 Harvard St. SE, Minneapolis, Minnesota 55455-0343, and Department of Psychiatry and Behavioral Neuroscience, McMaster University, 1200 Main St. West, Hamilton, Ontario L8N 2Z5, Canada

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm050644n

Reference30 articles.

1. Interaction of l-Prolyl-l-Leucyl Glycinamide with Dopamine D2Receptor: Evidence for Modulation of Agonist Affinity States in Bovine Striatal Membranes

2. Effects of prolyl-leucyl-glycinamide and cyclo(leucyl-glycine) on the supersensitivity of dopamine receptors in brain induced by chronic administration of haloperidol to rats

3. Potentiation of apomorphine action in rats by l-prolyl-l-leucyl-glycine amide

4. Modulation of Agonist Binding to Human Dopamine Receptor Subtypes by l-Prolyl-l-leucyl-glycinamide and a Peptidomimetic Analog

Cited by 33 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Allosteric Modulators of Dopamine D2 Receptors for Fine-Tuning of Dopaminergic Neurotransmission in CNS Diseases: Overview, Pharmacology, Structural Aspects and Synthesis;Molecules;2022-12-25

2. Exploring the role of neuropeptides in depression and anxiety;Progress in Neuro-Psychopharmacology and Biological Psychiatry;2022-03

3. A Convenient On-Site Oxidation Strategy for the N-Hydroxylation of Melanostatin Neuropeptide Using Cope Elimination;Synthesis;2021-11-11

4. Wandering beyond small molecules: peptides as allosteric protein modulators;Trends in Pharmacological Sciences;2021-11

5. Discovery of New Potent Positive Allosteric Modulators of Dopamine D2 Receptors: Insights into the Bioisosteric Replacement of Proline to 3-Furoic Acid in the Melanostatin Neuropeptide;Journal of Medicinal Chemistry;2021-04-16