Facile Radiosynthesis of Fluorine-18 Labeled β-Blockers. Synthesis, Radiolabeling, and ex Vivo Biodistribution of [18F]-(2S and 2R)-1-(1-Fluoropropan-2-ylamino)-3-(m-tolyloxy)propan-2-ol-Reference-Cited by-同舟云学术

Facile Radiosynthesis of Fluorine-18 Labeled β-Blockers. Synthesis, Radiolabeling, and ex Vivo Biodistribution of [18F]-(2S and 2R)-1-(1-Fluoropropan-2-ylamino)-3-(m-tolyloxy)propan-2-ol

Published:2008-07-26 Issue:16 Volume:51 Page:5093-5100
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Stephenson Karin A.¹,Wilson Alan A.¹,Meyer Jeffrey H.¹,Houle Sylvain¹,Vasdev Neil¹

Affiliation:

1. Centre for Addiction and Mental Health, 250 College Street, Toronto, Ontario, M5T 1R8 Canada, and Department of Psychiatry, University of Toronto, 250 College Street, Toronto, Ontario, M5T 1R8, Canada

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800227h

Reference36 articles.

1. PET Imaging of Beta-Adrenoceptors in Human Brain: A Realistic Goal or a Mirage?

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3. Effects of reboxetine and sertraline treatments alone and in combination on the binding properties of cortical NMDA and β1-adrenergic receptors in an animal model of depression

4. The effect of chronic administration of amitriptyline on the effects of subsequent electroconvulsive treatment on responsiveness of ?1- and ?-adrenoceptors in the rat cortical slices

5. Non-Invasive Molecular Imaging of β-Adrenoceptors In Vivo: Perspectives for PET-Radioligands

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