Bisoprolol-based 18F-PET tracer: Synthesis and preliminary in vivo validation of β1-blocker selectivity for β1-adrenergic receptors in the heart

Author:

Kang Julie,More Kunal N.,Pyo Ayoung,Jung Yerim,Kim Dong-Yeon,Chang Dong-Jo

Funder

National Research Foundation of Korea

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference28 articles.

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3. The pharmacological specificity of beta-1 and beta-2 adrenergic receptors in rat heart and lung in vitro;Mineman;Mol Pharmacol,1979

4. β-Adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177;De Paermentier;Eur J Pharmacol,1989

5. Pharmacotherapeutics for advanced practice: a practical approach;Arcangelo,2006

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