Indolylarylsulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: New Cyclic Substituents at Indole-2-carboxamide

Author:

La Regina Giuseppe1,Coluccia Antonio1,Brancale Andrea2,Piscitelli Francesco1,Gatti Valerio1,Maga Giovanni3,Samuele Alberta3,Pannecouque Christophe4,Schols Dominique4,Balzarini Jan4,Novellino Ettore5,Silvestri Romano1

Affiliation:

1. Istituto Pasteur - Fondazione Cenci Bolognetti, Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, Piazzale Aldo Moro 5, I-00185 Roma, Italy

2. Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3NB, U.K.

3. Istituto di Genetica Molecolare, Consiglio Nazionale delle Ricerche, Via Abbiategrasso 207, I-27100 Pavia, Italy

4. Rega Institute for Medical Research, Katholieke Universiteit Leuven, B-3000 Leuven, Belgium

5. Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli Federico II, Via Domenico Montesano 49, I-80131, Napoli, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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