Impact of Radiolabeling Strategies on the Pharmacokinetics and Distribution of an Anti-PD-L1 PET Ligand-Reference-Cited by-同舟云学术

Impact of Radiolabeling Strategies on the Pharmacokinetics and Distribution of an Anti-PD-L1 PET Ligand

Published:2022-08-23 Issue:10 Volume:19 Page:3673-3680
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Tran Vu Long¹,Bouleau Alizée¹,Nozach Hervé²,Richard Mylène¹,Chevaleyre Céline¹,Dubois Steven²,Kereselidze Dimitri¹,Kuhnast Bertrand¹^ORCID,Evans Michael J.³^ORCID,Specklin Simon¹^ORCID,Truillet Charles¹^ORCID

Affiliation:

1. Université Paris-Saclay, CEA, CNRS, Inserm, BioMaps, SHFJ, Orsay 91400, France

2. Université Paris-Saclay, CEA, DMTS, SIMoS, CEA-Saclay, Gif-sur-Yvette CEDEX 91191, France

3. Department of Radiology and Biomedical Imaging, UCSF, San Francisco, California 94107, United States

Funder

Agence Nationale de la Recherche

Fondation ARC pour la Recherche sur le Cancer

National Institute of Biomedical Imaging and Bioengineering

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.molpharmaceut.2c00497

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4. Molecular Imaging of PD-L1 Expression and Dynamics with the Adnectin-Based PET Tracer 18F-BMS-986192

5. Synthesis and Biologic Evaluation of a Novel 18F-Labeled Adnectin as a PET Radioligand for Imaging PD-L1 Expression

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