Process Improvements for the Manufacture of Tenofovir Disoproxil Fumarate at Commercial Scale-Reference-Cited by-同舟云学术

Process Improvements for the Manufacture of Tenofovir Disoproxil Fumarate at Commercial Scale

Published:2010-08-24 Issue:5 Volume:14 Page:1194-1201
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Brown Ripin David H.¹,Teager David S.¹,Fortunak Joseph¹,Basha Shaik Mahaboob¹,Bivins Nylea¹,Boddy Christopher N.¹,Byrn Stephen¹,Catlin Kelly K.¹,Houghton Stephen R.¹,Jagadeesh S. Tirumala¹,Kumar K. Anesh¹,Melton Jack¹,Muneer Shaik¹,Rao L. Nagaprasada¹,Rao R. Venkateswara¹,Ray Puma Chandra¹,Reddy Nardla Gopal¹,Reddy Ravi Mallikarjuna¹,Shekar K. Chandra¹,Silverton Tricia¹,Smith Daniel T.¹,Stringham Rodger W.¹,Subbaraju Gottumukkala V.¹,Talley Frajovon¹,Williams Adrian¹

Affiliation:

1. Clinton Health Access Initiative, 383 Dorchester Avenue, Suite 400, Boston, Massachusetts 02127, U.S.A., Department of Chemistry, Howard University, 525 College Street NW, Washington, D.C. 20059, U.S.A., Department of Chemistry, University of Ottawa, Ottawa, Ontario ON K1N 6N5, Canada, Department of Industrial and Physical Pharmacy, Purdue University, 575 Stadium Mall Drive, West Lafayette, Indiana 47907-2091, U.S.A., ProcesScience, Inc., 117 Woodberry Lane, Fayetteville, New York 13066, U.S.A., Inogent...

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op1001337

Reference13 articles.

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3. Anti-Human Immunodeficiency Virus Activity and Cellular Metabolism of a Potential Prodrug of the Acyclic Nucleoside Phosphonate 9- R -(2-Phosphonomethoxypropyl)adenine (PMPA), Bis(isopropyloxymethylcarbonyl)PMPA

4. Differential antiherpesvirus and antiretrovirus effects of the (S) and (R) enantiomers of acyclic nucleoside phosphonates: potent and selective in vitro and in vivo antiretrovirus activities of (R)-9-(2-phosphonomethoxypropyl)-2,6-diaminopurine

5. Arimilli, M. N.; Cundy, K. C.; Dougherty, J. P.; Kim, C. U.; Oliyai, R.; Stella, V. J.U.S. Patent 5,922,695, 1998.

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