Development of a Large-Scale Copper(I)/TEMPO-Catalyzed Aerobic Alcohol Oxidation for the Synthesis of LSD1 Inhibitor GSK2879552-Reference-Cited by-同舟云学术

Development of a Large-Scale Copper(I)/TEMPO-Catalyzed Aerobic Alcohol Oxidation for the Synthesis of LSD1 Inhibitor GSK2879552

Published:2018-10-25 Issue:1 Volume:38 Page:176-184
ISSN:0276-7333
Container-title:Organometallics
language:en
Short-container-title:Organometallics

Author:

Ochen Augustine,Whitten Robert,Aylott Helen E.,Ruffell Katie,Williams Glynn D.,Slater Fiona,Roberts Andrew,Evans Paul,Steves Janelle E.¹^ORCID,Sanganee Mahesh J.

Affiliation:

1. API Chemistry, GlaxoSmithKline, 1250 South Collegeville Rd., Collegeville, Pennsylvania 19426, United States

Publisher

American Chemical Society (ACS)

Subject

Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.organomet.8b00546

Reference53 articles.

1. Activated Dimethyl Sulfoxide: Useful Reagents for Synthesis

2. Readily accessible 12-I-5 oxidant for the conversion of primary and secondary alcohols to aldehydes and ketones

3. Analysis of the reactions used for the preparation of drug candidate molecules

4. A Scalable Oxidation for the Final Stage of Synthesis of Cathepsin K Inhibitor SB-462795

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