Discovery of a Novel Class of Substituted Pyrrolooctahydroisoquinolines as Potent and Selective δ Opioid Agonists, Based on an Extension of the Message−Address Concept-Reference-Cited by-同舟云学术

Discovery of a Novel Class of Substituted Pyrrolooctahydroisoquinolines as Potent and Selective δ Opioid Agonists, Based on an Extension of the Message−Address Concept

Published:1997-09-01 Issue:20 Volume:40 Page:3192-3198
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Dondio Giulio¹,Ronzoni Silvano¹,Eggleston Drake S.¹,Artico Marco¹,Petrillo Paola¹,Petrone Giuseppe¹,Visentin Luciano¹,Farina Carlo¹,Vecchietti Vittorio¹,Clarke Geoffrey D.¹

Affiliation:

1. SmithKline Beecham S.p.A., Via Zambeletti, 20021 Baranzate, Milan, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9608218

Reference32 articles.

1. κ-Opioid receptors and analgesia

2. Opioid-induced stimulation of fetal respiratory activity by [D-Ala2]deltorphin I

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