Cyclic Enkephalins with a Diversely Substituted Guanidine Bridge or a Thiourea Bridge: Synthesis, Biological and Structural Evaluations-Reference-Cited by-同舟云学术

Cyclic Enkephalins with a Diversely Substituted Guanidine Bridge or a Thiourea Bridge: Synthesis, Biological and Structural Evaluations

Published:2013-07-12 Issue:14 Volume:56 Page:5964-5973
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Touati-Jallabe Youness¹,Bojnik Engin²,Legrand Baptiste³,Mauchauffée Elodie¹,Chung Nga N.⁴,Schiller Peter W.⁴⁵,Benyhe Sandor²,Averlant-Petit Marie-Christine³,Martinez Jean¹,Hernandez Jean-François¹

Affiliation:

1. Institut des Biomolécules Max Mousseron, CNRS UMR 5247, Université Montpellier 1, Université Montpellier 2, Faculté de Pharmacie, 15 Avenue Charles Flahault, 34093 Montpellier cedex 05, France

2. Biological Research Center, Institute of Biochemistry, POB 521, H-6702 Szeged, Hungary

3. Laboratoire de Chimie Physique Macromoléculaire, CNRS UMR 7568, Université de Lorraine, 1 rue Grandville, 54001 Nancy Cedex, France

4. Laboratory of Chemical Biology and Peptide Research, Clinical Research Institute of Montreal, 110 Pine Avenue West, Montreal, Quebec H2W 1R7, Canada

5. Department of Pharmacology, Université de Montréal, Montreal, Quebec H3C 3J7, Canada

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm4008592

Reference32 articles.

1. Cyclic Peptides with a Diversely Substituted Guanidine Bridge: Solid-Phase Synthesis and Structural Analysis

2. Identification of two related pentapeptides from the brain with potent opiate agonist activity

3. Development and validation of opioid ligand-receptor interaction models: The structural basis of mu vs. delta selectivity

4. Conformation-activity relationships of opioid peptides with selective activities at opioid receptors

5. Use of NMR and Fluorescence Spectroscopy as well as Theoretical Conformational Analysis in Conformation-activity Studies of Cyclic Enkephalin Analogues

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