Development and validation of opioid ligand-receptor interaction models: The structural basis of mu vs. delta selectivity
Author:
Publisher
Wiley
Subject
Endocrinology,Biochemistry
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1034/j.1399-3011.2002.21061.x/fullpdf
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3. Conformational analysis of the δ receptor-selective, cyclic opioid peptide, Tyr-c[d-Cys-Phe-d-Pen]OH (JOM-13). Comparison of X-ray crystallographic structures, molecular mechanics simulations and 1H NMR data;Lomize;J. Am. Chem. Soc.,1994
4. Development of a model for the δ opioid receptor pharmacophore. 1. Conformationally restricted Tyr1 replacements in the cyclic δ receptor selective tetrapeptide Tyr-c[d-Cys-Phe-d-Pen]OH (JOM-13);Mosberg;J. Med. Chem.,1994
5. Development of a model for the δ opioid receptor pharmacophore. 2. Conformationally restricted Phe3 replacements in the cyclic δ receptor selective tetrapeptide Tyr-c[d-Cys-Phe-d-Pen]OH (JOM-13);Mosberg;J. Med. Chem.,1994
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