2(S)-((3,5-Bis(trifluoromethyl)benzyl)oxy)-3(S)-phenyl-4-((3-oxo-1,2,4-triazol- 5-yl)methyl)morpholine (1): A Potent, Orally Active, Morpholine-Based Human Neurokinin-1 Receptor Antagonist-Reference-Cited by-同舟云学术

2(S)-((3,5-Bis(trifluoromethyl)benzyl)oxy)-3(S)-phenyl-4-((3-oxo-1,2,4-triazol- 5-yl)methyl)morpholine (1): A Potent, Orally Active, Morpholine-Based Human Neurokinin-1 Receptor Antagonist

Published:1996-01-01 Issue:9 Volume:39 Page:1760-1762
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hale Jeffrey J.¹,Mills Sander G.¹,MacCoss Malcolm¹,Shah Shrenik K.¹,Qi Hongbo¹,Mathre David J.¹,Cascieri Margaret A.¹,Sadowski Sharon¹,Strader Catherine D.¹,MacIntyre D. Euan¹,Metzger Joseph M.¹

Affiliation:

1. Merck Research Laboratories, Rahway, New Jersey 07065

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm950654w

Reference33 articles.

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