Preparation of the HIV Attachment Inhibitor BMS-663068. Part 4. Synthesis of the 6-Azaindole Core-Reference-Cited by-同舟云学术

Preparation of the HIV Attachment Inhibitor BMS-663068. Part 4. Synthesis of the 6-Azaindole Core

Published:2017-08-09 Issue:8 Volume:21 Page:1131-1136
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Bultman Michael S.¹^ORCID,Fan Junying¹,Fanfair Dayne¹,Soltani Michelle¹,Simpson James¹,Murugesan Saravanababu¹,Soumeillant Maxime¹,Chen Ke¹,Risatti Christina¹,La Cruz Thomas E.¹^ORCID,Buono Frederic G.¹,Hung Victor¹,Schild Richard L.¹,Ivy Sabrina¹,Sweeney Jason T.¹,Conlon David A.¹,Eastgate Martin D.¹^ORCID

Affiliation:

1. Chemical & Synthetic Development, Bristol-Myers Squibb Company, One Squibb Drive, New Brunswick, New Jersey, 08903-0191, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.7b00152

Reference19 articles.

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3. Novel indole and azaindole (pyrrolopyridine) cannabinoid (CB) receptor agonists: Design, synthesis, structure–activity relationships, physicochemical properties and biological activity

4. Novel 3-Azaindolyl-4-arylmaleimides Exhibiting Potent Antiangiogenic Efficacy, Protein Kinase Inhibition, and Antiproliferative Activity

5. Site-Selective Azaindole Arylation at the Azine and Azole Rings via N-Oxide Activation

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