Scale-Up Synthesis of IID572: A New β-Lactamase Inhibitor-Reference-Cited by-同舟云学术

Scale-Up Synthesis of IID572: A New β-Lactamase Inhibitor

Published:2020-05-14 Issue:7 Volume:24 Page:1244-1253
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Furegati Markus¹^ORCID,Nocito Sandro¹,Reck Folkert²^ORCID,Casarez Anthony²,Simmons Robert²,Schuetz Heiner¹,Koch Guido¹

Affiliation:

1. Synthesis and Technologies Group, Novartis Institutes for BioMedical Research, Klybeckstrasse 141, Basel 4057, Switzerland

2. Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, California 94608, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.0c00069

Reference19 articles.

1. IID572: A New Potentially Best-In-Class β-Lactamase Inhibitor

2. Ronsheim, M. S.; Racha, S.; Lawton, G. R.; Zhou, S. H.; Kalyan, Y. B.; Golden, M.; Milne, D.; Telford, A.; Cherryman, J.; Boyd, A.; Phillips, A. J.; Dedhiya, M. G. Processes for Preparing Heterocyclic Compounds Including Trans-7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide and Salts Thereof. US2,012,323,010, 2012.

3. Development of a Manufacturing Route to Avibactam, a β-Lactamase Inhibitor

4. Carboxylic Acids as A Traceless Activation Group for Conjugate Additions: A Three-Step Synthesis of (±)-Pregabalin

5. [4 + 2]-Cycloadditionen von ?,?-unges�ttigten Hydrazonen. Teil 1. Pyridin-2,3-dicarboximide aus 1-(Dimethylamino)-1,4-dihydropyridin-Derivaten

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