Facile and Cost-Effective Route for the Synthesis of Simmerafil-Reference-Cited by-同舟云学术

Facile and Cost-Effective Route for the Synthesis of Simmerafil

Published:2021-10-19 Issue:11 Volume:25 Page:2432-2437
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Odilov Abdullajon¹²,Liu Yin¹²,Hu Tianwen²³,Jiang Xiangrui¹²^ORCID,Suo Jin¹,Tian Guanghui⁴,Yang Feipu¹^ORCID,Shen Jingshan¹²^ORCID

Affiliation:

1. CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, P. R. China

2. University of Chinese Academy of Sciences, Beijing 100049, P. R. China

3. Key Laboratory of Plant Resources and Chemistry in Arid Regions, Xinjiang Technical Institute of Physics and Chemistry, Chinese Academy of Sciences, Urumqi 830011, Xinjiang, P. R. China

4. Vigonvita Life Science Co., Ltd., Suzhou, Jiangsu 215123, P. R. China

Funder

Ministry of Science and Technology of the People's Republic of China

National Science and Technology Major Project

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.1c00184

Reference13 articles.

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2. Targeted Drugs for Treatment of Pulmonary Arterial Hypertension: Past, Present, and Future Perspectives

3. Liu, Z.; Li, J. F.; Yang, X. J.; Wang, Z.; Zhang, J. F.; Zhu, Y.; Tian, G. H.; Jin, Q.; Shen, J. K.; Zhu, W. L.; Phenyl pyrimidone compounds, pharmaceutical compositions, preparation methods and uses thereof. EP2383262A1, 2011.

4. Shen, J. S.; He, Y.; Chen, W. M.; Li, J. F.; Tian, G. H.; Gong, X. D.; Wang, Z.; Zhang, R. X.; Liu, Y. J.; Jiang, H. L. Salt and polymorph of benzopyrimidinone compound and pharmaceutical composition and use thereof. US2020,140,415A1, 2020.

5. Radiosynthesis of a carbon-11 labeled PDE5 inhibitor [11C]TPN171 as a new potential PET heart imaging agent

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