Practical and Efficient Synthesis of 2-Thio-imidazole Derivative—ZY12201: A Potent TGR5 Agonist-Reference-Cited by-同舟云学术

登录注册会员服务联系我们

Practical and Efficient Synthesis of 2-Thio-imidazole Derivative—ZY12201: A Potent TGR5 Agonist

Published:2020-07-30 Issue:8 Volume:24 Page:1508-1514
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Joshi Vivek M.¹²,Sojitra Chandrakant¹²³,Sasane Santosh¹²,Shukla Mrigendra¹,Chauhan Rakesh¹,Chaubey Vipin¹,Jain Sarika¹,Shah Kalpesh¹,Mande Hemant²,Soman Shubhangi²,Pamidimukkala Padmaja Sudhakar²^ORCID,Shah Shailesh R.²^ORCID,Pandey Bipin¹,Singh Kumar K.³,Agarwal Sameer¹^ORCID

Affiliation:

1. Zydus Research Centre, Cadila Healthcare Ltd., Sarkhej-Bavla N.H. No. 8 A, Moraiya, Ahmedabad 382210, India

2. Department of Chemistry, Faculty of Science, M. S. University of Baroda, Baroda 390002, India

3. API Division, Cadila Healthcare Limited, Sarkhej-Bavla N.H. No. 8 A, Changodar, Ahmedabad 382210, India

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.0c00234

Reference20 articles.

1. Diabesity: an overview of a rising epidemic

2. Pharmacological Agents That Directly Modulate Insulin Secretion

3. Non-insulin therapies for type 2 diabetes

4. Identification of an Orally Efficacious GPR40/FFAR1 Receptor Agonist

Cited by 4 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Mechanism of action of the bile acid receptor TGR5 in obesity;Acta Pharmaceutica Sinica B;2024-02

2. ZY12201: A Potent TGR5 Agonist: Identification of a Novel Pan CYP450 Inhibitor Tool Compound for In-Vitro Assessment;Drug Metabolism and Bioanalysis Letters;2022-07

3. Multigram-scale synthesis of GSK 2,256,294, an inhibitor of soluble epoxide hydrolase in clinical evaluation;Chemical Papers;2022-01-20

4. Identification of degradation impurity of TGR5 receptor agonist-ZY12201 by LC–MS technique during force degradation study;SN Applied Sciences;2021-05-25

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号京ICP备18003416号-3