A Practical and Scalable Method for Manufacturing JAK Inhibitor ASP3627
Author:
Affiliation:
1. Process Chemistry Labs., Pharmaceutical Technology, Astellas Pharma Inc., 160-2 Akahama, Takahagi-shi, Ibaraki 318-0001, Japan
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.9b00269
Reference27 articles.
1. JAK inhibition as a therapeutic strategy for immune and inflammatory diseases
2. Tofacitinib Synthesis – An Asymmetric Challenge
3. An Improved and Efficient Process for the Preparation of Tofacitinib Citrate
4. Solution-Phase Parallel Synthesis of Ruxolitinib-Derived Janus Kinase Inhibitors via Copper-Catalyzed Azide–Alkyne Cycloaddition
5. Enantioselective Synthesis of Janus Kinase Inhibitor INCB018424 via an Organocatalytic Aza-Michael Reaction
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