An Improved and Efficient Process for the Preparation of Tofacitinib Citrate-Reference-Cited by-同舟云学术

An Improved and Efficient Process for the Preparation of Tofacitinib Citrate

Published:2014-11-21 Issue:12 Volume:18 Page:1714-1720
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Patil Yogesh S.¹,Bonde Nilesh L.¹,Kekan Ankush S.¹,Sathe Dhananjay G.¹,Das Arijit¹

Affiliation:

1. Unichem Laboratories Limited, Center of Excellence, Process Research, Pilerne Industrial Estate, Plot No-12 to 16, Pilerne, Bardez, Goa 403511, India

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op500274j

Reference13 articles.

1. aBlumenkopf, T. A.; Flanagan, M. E.; Munchhof, M. J.U.S. Patent USRE41783E, 2010.

2. bFlanagan, M. E.; Munchhof, M. J.U.S. Patent US7301023B2, 2007.

3. cErnest, W. G.; Christian, K.; Ton, V.; Edward, F. M.; Munchhof, M. J.PCT WO 02096909, 2002.

4. Asymmetric total synthesis of Tofacitinib

5. bStavber, G.; Cluzean, J.PCT WO 2014016338A1, 2014.

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