Use of Phosphazene Base BTPP for Phosphorylative Activation in the Scale-Up of BET Inhibitor GSK525762-Reference-Cited by-同舟云学术

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Use of Phosphazene Base BTPP for Phosphorylative Activation in the Scale-Up of BET Inhibitor GSK525762

Published:2022-08-18 Issue:9 Volume:26 Page:2646-2655
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Jones Rhiannon E. H.¹^ORCID,Aspin Peter¹,Davies Suzanne H.¹,Mann Inderjit¹,Priestley Catherine¹,Roberts Andrew D.¹,Zotova-Eldridge Natalia¹,Leahy John H.¹

Affiliation:

1. Medicinal Science and Technology, GlaxoSmithKline Medicines Research Centre, Stevenage SG1 2NY, U.K.

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.2c00048

Reference25 articles.

1. Selective inhibition of BET bromodomains

2. Discovery and Characterization of Small Molecule Inhibitors of the BET Family Bromodomains

3. Suppression of inflammation by a synthetic histone mimic

4. Abstract 4693: Mechanism-based combination strategies for BET inhibitors in NUT midline carcinoma

5. Discovery of Epigenetic Regulator I-BET762: Lead Optimization to Afford a Clinical Candidate Inhibitor of the BET Bromodomains

Cited by 1 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. A strategy for the controllable generation of organic superbases from benchtop-stable salts;Chemical Science;2024

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