Discovery and Characterization of Small Molecule Inhibitors of the BET Family Bromodomains-Reference-Cited by-同舟云学术

Discovery and Characterization of Small Molecule Inhibitors of the BET Family Bromodomains

Published:2011-05-13 Issue:11 Volume:54 Page:3827-3838
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Chung Chun-wa¹,Coste Hervé²,White Julia H.¹,Mirguet Olivier²,Wilde Jonathan¹,Gosmini Romain L.²,Delves Chris¹,Magny Sylvie M.²,Woodward Robert¹,Hughes Stephen A.¹,Boursier Eric V.²,Flynn Helen¹,Bouillot Anne M.²,Bamborough Paul¹,Brusq Jean-Marie G.²,Gellibert Françoise J.²,Jones Emma J.¹,Riou Alizon M.²,Homes Paul¹,Martin Sandrine L.²,Uings Iain J.³,Toum Jérôme²,Clément Catherine A.²,Boullay Anne-Bénédicte²,Grimley Rachel L.¹,Blandel Florence M.²,Prinjha Rab K.³,Lee Kevin³,Kirilovsky Jorge²,Nicodeme Edwige²

Affiliation:

1. Molecular Discovery Research, GlaxoSmithKline R&D, Stevenage SG5 4HT, U.K.

2. Lipid Metabolism Discovery Performance Unit, GlaxoSmithKline R&D, Les Ulis, France

3. Epinova, Discovery Performance Unit, GlaxoSmithKline R&D, Stevenage SG5 4HT, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200108t

Reference34 articles.

1. Epigenetics: A Landscape Takes Shape