Review of Synthetic Routes and Crystalline Forms of the Antiandrogen Oncology Drugs Enzalutamide, Apalutamide, and Darolutamide

Author:

Hughes David L.1ORCID

Affiliation:

1. Cidara Therapeutics, 6310 Nancy Ridge Drive, Suite 101, San Diego, California 92121, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Reference93 articles.

1. Development of a Second-Generation Antiandrogen for Treatment of Advanced Prostate Cancer

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3. aSawyers, C. L.; Jung, M. E.; Chen, C. D.; Ouk, S.; Welsbie, D.; Tran, C.; Wongvipat, J.; Yoo, D. Diarylhydantoin Compounds. PCT Int. Patent Appl. WO 2006/124118, November 23, 2006.

4. bSawyers, C. L.; Jung, M. E.; Chen, C. D.; Ouk, S.; Welsbie, D.; Tran, C.; Wongvipat, J.; Yoo, D. Diarylhydantoin Compounds. U.S. Patent 7709517 B2, May 4, 2010.

5. cJung, M. E.; Yoo, D.; Sawyers, C. L.; Tran, C.; Wongvipat, J. Diarylhydantoin Compounds. U.S. Patent 8110594 B2, February 7, 2012.

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