Large Scale Synthesis of an Ampakine-type Active Pharmaceutical Ingredient Based on a Telescoped Regioselective Double Amidation Reaction-Reference-Cited by-同舟云学术

Large Scale Synthesis of an Ampakine-type Active Pharmaceutical Ingredient Based on a Telescoped Regioselective Double Amidation Reaction

Published:2019-07-11 Issue:9 Volume:23 Page:1932-1947
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Hardouin Christophe¹^ORCID,Pin Frédéric¹,Giffard Jean-François¹,Hervouet Yvon¹,Hublet Julie¹,Janvier Solenn¹,Penloup Christine¹,Picard Julien¹,Pinault Nathalie¹,Schiavi Bruno¹,Zhang Peng²,Zhao Weiwei²,Zhu Xueyan²

Affiliation:

1. Industrial Research Centre, Oril Industrie, 13 rue Desgenétais, 76210 Bolbec, France

2. Shanghai Institute of Pharmaceutical Indus China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Pudong District, Shanghai 201203, People’s Republic of China

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.9b00241

Reference30 articles.

1. Ligands for Glutamate Receptors: Design and Therapeutic Prospects

2. Glutamate Receptor Ion Channels: Structure, Regulation, and Function

3. Distribution of [3H]AMPA binding sites in rat brain as determined by quantitative autoradiography

4. Learning Induces Long-Term Potentiation in the Hippocampus

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