Design and Synthesis of Potent and Selective α4β7 Integrin Antagonists-Reference-Cited by-同舟云学术

Design and Synthesis of Potent and Selective α4β7 Integrin Antagonists

Published:2001-07-26 Issue:16 Volume:44 Page:2586-2592
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Boer Jürgen¹,Gottschling Dirk¹,Schuster Anja¹,Semmrich Monika¹,Holzmann Bernhard¹,Kessler Horst¹

Affiliation:

1. Institut für Organische Chemie und Biochemie, Technische Universität München, Lichtenbergstrasse 4, D-85747 Garching, Germany, and Institut für Medizinische Mikrobiologie, Immunologie und Hygiene, Technische Universität München, Trogerstrasse 4a, D-81675 München, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0005508

Reference49 articles.

1. Integrins: Versatility, modulation, and signaling in cell adhesion

2. Eble, J. A. Integrins − a versatile and old family of cell adhesion molecules.Integrin-Ligand Interaction; Springer-Verlag: Heidelberg, 1997; pp 1−40.

3. VLA Proteins in the Integrin Family: Structures, Functions, and Their Role on Leukocytes

4. α4β7 integrin mediates lymphocyte binding to the mucosal vascular addressin MAdCAM-1

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