SAR Development of Lysine-Based Irreversible Inhibitors of Transglutaminase 2 for Huntington's Disease-Reference-Cited by-同舟云学术

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SAR Development of Lysine-Based Irreversible Inhibitors of Transglutaminase 2 for Huntington's Disease

Published:2012-10-08 Issue:12 Volume:3 Page:1024-1028
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Wityak John¹,Prime Michael E.²,Brookfield Frederick A.²,Courtney Stephen M.²,Erfan Sayeh²,Johnsen Siw²,Johnson Peter D.²,Li Marie²,Marston Richard W.²,Reed Laura²,Vaidya Darshan²,Schaertl Sabine³,Pedret-Dunn Anna²,Beconi Maria¹,Macdonald Douglas¹,Muñoz-Sanjuan Ignacio¹,Dominguez Celia¹

Affiliation:

1. CHDI Management/CHDI Foundation, 6080 Center Drive, Suite 100, Los Angeles, California 90045, United States

2. Evotec (U.K.) Ltd., 114 Milton Park, Abingdon, OX14 4SA, United Kingdom

3. Evotec AG, Manfred Eigen Campus, Essener Bogen 7, 22419 Hamburg, Germany

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml300241m

Reference25 articles.

1. Transglutaminases: multifunctional cross‐linking enzymes that stabilize tissues

2. Regulation of Human Tissue Transglutaminase Function by Magnesium-Nucleotide Complexes

3. A novel function of tissue-type transglutaminase: protein disulphide isomerase

4. Transglutaminase 2 Undergoes a Large Conformational Change upon Activation

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1. Preclinical evaluation of an 18F-labeled Nε-acryloyllysine piperazide for covalent targeting of transglutaminase 2;EJNMMI Radiopharmacy and Chemistry;2024-01-02

2. Discovery and Characterization of PROTACs Targeting Tissue Transglutaminase (TG2);Journal of Medicinal Chemistry;2023-07-14

3. Novel irreversible peptidic inhibitors of transglutaminase 2;RSC Medicinal Chemistry;2023

4. The Emerging Landscape of Small-Molecule Therapeutics for the Treatment of Huntington’s Disease;Journal of Medicinal Chemistry;2022-12-09

5. Application of a Fluorescence Anisotropy-Based Assay to Quantify Transglutaminase 2 Activity in Cell Lysates;International Journal of Molecular Sciences;2022-04-19

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