(Heteroarylmethyl)benzoic Acids as a New Class of Bacterial Cystathionine γ-Lyase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling-Reference-Cited by-同舟云学术

(Heteroarylmethyl)benzoic Acids as a New Class of Bacterial Cystathionine γ-Lyase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling

Published:2024-05-21 Issue:6 Volume:10 Page:2127-2150
ISSN:2373-8227
Container-title:ACS Infectious Diseases
language:en
Short-container-title:ACS Infect. Dis.

Author:

Golovina Anastasia¹^ORCID,Proia Eleonora²,Fiorentino Francesco³^ORCID,Yunin Maxim¹^ORCID,Kasatkina Maria¹,Zigangirova Nailya⁴,Soloveva Anna⁴,Sysolyatina Elena⁴,Ermolaeva Svetlana⁴,Novikov Roman⁵^ORCID,Silonov Sergei¹⁶,Pushkin Sergei¹,Mladenović Milan⁷^ORCID,Isakova Julia¹,Belik Albina¹,Nawrozkij Maxim¹,Rotili Dante³^ORCID,Ragno Rino²^ORCID,Ivanov Roman¹

Affiliation:

1. Sirius University of Science and Technology, Olympic Avenue, 1, Sirius , Krasnodar Region 354340, Russia

2. Rome Center for Molecular Design, Department of Drug Chemistry and Technologies, Sapienza University of Rome, P. le A. Moro 5 , Rome 00185, Italy

3. Department of Drug Chemistry and Technologies, Sapienza University of Rome, P. le A. Moro 5, Rome 00185, Italy

4. National Research Centre of Epidemiology and Microbiology named after N. F. Gamaleya, Russian Health Ministry, Gamaleya St.18 , 123098 Moscow, Russia

5. Engelhardt Institute of Molecular Biology of the Russian Academy of Sciences, 32 Vavilov St. , Moscow 119991, Russia

6. Laboratory of Structural Dynamics, Stability and Folding of Proteins, Institute of Cytology, Russian Academy of Sciences, 4 Tikhoretsky Avenue , St. Petersburg 194064, Russia

7. Kragujevac Center for Computational Biochemistry, Department of Chemistry, Faculty of Science, University of Kragujevac, Radoja Domanovića 12 , Kragujevac 34000, P.O. Box 60, Serbia

Funder

European Commission

Sapienza Università di Roma

Ministry of Science and Higher Education of the Russian Federation

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acsinfecdis.4c00136

Reference36 articles.

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5. H2S as a Bacterial Defense Against Antibiotics