Structural Requirements for Dihydrobenzoxazepinone Anthelmintics: Actions against Medically Important and Model Parasites: Trichuris muris, Brugia malayi, Heligmosomoides polygyrus, and Schistosoma mansoni-Reference-Cited by-同舟云学术

Structural Requirements for Dihydrobenzoxazepinone Anthelmintics: Actions against Medically Important and Model Parasites: Trichuris muris, Brugia malayi, Heligmosomoides polygyrus, and Schistosoma mansoni

Published:2021-04-02 Issue:5 Volume:7 Page:1260-1274
ISSN:2373-8227
Container-title:ACS Infectious Diseases
language:en
Short-container-title:ACS Infect. Dis.

Author:

Partridge Frederick A.¹^ORCID,Bataille Carole J.R.²,Forman Ruth³,Marriott Amy E.⁴,Forde-Thomas Josephine⁵,Häberli Cécile⁶⁷,Dinsdale Ria L.²,O’Sullivan James D.B.³⁸,Willis Nicky J.²⁹,Wynne Graham M.²,Whiteland Helen⁵,Archer John⁴,Steven Andrew⁴,Keiser Jennifer⁶⁷,Turner Joseph D.⁴¹⁰,Hoffmann Karl F.⁵^ORCID,Taylor Mark J.⁴¹⁰,Else Kathryn J.³,Russell Angela J.²¹¹^ORCID,Sattelle David B.¹

Affiliation:

1. Centre for Respiratory Biology, UCL Respiratory, Division of Medicine, University College London, London WC1E 6JF, United Kingdom

2. Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Oxford OX1 3TA, United Kingdom

3. Lydia Becker Institute of Immunology and Inflammation, Faculty of Biology, Medicine and Health, University of Manchester, Manchester M13 9PT, United Kingdom

4. Centre for Drugs and Diagnostics, Department of Tropical Disease Biology, Liverpool School of Tropical Medicine, Liverpool L3 5QA, United Kingdom

5. Institute of Biological, Environmental and Rural Sciences (IBERS), Aberystwyth University, Aberystwyth, Wales SY23 3DA, United Kingdom

6. Department of Medical Parasitology and Infection Biology, Swiss Tropical and Public Health Institute, Socinstrasse 57, Basel CH-4002, Switzerland

7. University of Basel, Petersplatz 1, Basel CH-4001, Switzerland

8. Henry Royce Institute, The University of Manchester, Oxford Road, Manchester M13 9PL, United Kingdom

9. Alzheimer’s Research UK UCL Drug Discovery Institute, University College London, Gower Street, London WC1E 6BT, United Kingdom

10. Centre for Neglected Tropical Diseases, Liverpool School of Tropical Medicine, Liverpool L3 5QA, United Kingdom

11. Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, United Kingdom

Funder

Research Councils UK

University of Manchester

Bill and Melinda Gates Foundation

National Centre for the Replacement Refinement and Reduction of Animals in Research

Wellcome Trust

University College London

Welsh Government Life Sciences Research Network Wales

Publisher

American Chemical Society (ACS)

Subject

Infectious Diseases

Link

https://pubs.acs.org/doi/pdf/10.1021/acsinfecdis.1c00025

Reference76 articles.

1. Global, regional, and national incidence, prevalence, and years lived with disability for 354 diseases and injuries for 195 countries and territories, 1990–2017: a systematic analysis for the Global Burden of Disease Study 2017

2. Global, regional, and national disability-adjusted life-years (DALYs) for 359 diseases and injuries and healthy life expectancy (HALE) for 195 countries and territories, 1990–2017: a systematic analysis for the Global Burden of Disease Study 2017

3. World Health Organization. (2020) 2030 Targets for Soil-Transmitted Helminthiases Control Programmes.

4. Efficacy and Safety of a Single Dose versus a Multiple Dose Regimen of Mebendazole against Hookworm Infections in Children: A Randomised, Double-blind Trial

5. Efficacy of Current Drugs Against Soil-Transmitted Helminth Infections

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