Challenges in the Development of a Thiol-Based Broad-Spectrum Inhibitor for Metallo-β-Lactamases-Reference-Cited by-同舟云学术

Challenges in the Development of a Thiol-Based Broad-Spectrum Inhibitor for Metallo-β-Lactamases

Published:2017-11-26 Issue:3 Volume:4 Page:360-372
ISSN:2373-8227
Container-title:ACS Infectious Diseases
language:en
Short-container-title:ACS Infect. Dis.

Author:

Büttner Dominik,Kramer Jan S.,Klingler Franca-M.,Wittmann Sandra K.,Hartmann Markus R.,Kurz Christian G.,Kohnhäuser Daniel,Weizel Lilia,Brüggerhoff Astrid,Frank Denia¹,Steinhilber Dieter,Wichelhaus Thomas A.¹,Pogoryelov Denys,Proschak Ewgenij^ORCID

Affiliation:

1. Institute of Medical Microbiology and Infection Control, Goethe University Hospital, Paul-Ehrlich-Straße 40, 60596 Frankfurt, Germany

Funder

Deutsche Forschungsgemeinschaft

Publisher

American Chemical Society (ACS)

Subject

Infectious Diseases

Link

https://pubs.acs.org/doi/pdf/10.1021/acsinfecdis.7b00129

Reference45 articles.

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2. WHO (2014) Antibiotic Resistance Global Report on Surveillance, http://apps.who.int/iris/bitstream/10665/112642/1/9789241564748_eng.pdf (accessed Aug 03 2017).

3. Structure of New Delhi metallo-β-lactamase 1 (NDM-1)

4. ESKAPEing the labyrinth of antibacterial discovery

5. The Challenge of Overcoming Antibiotic Resistance: An Adjuvant Approach?

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