A Chemical Switch for the Modulation of the Functional Activity of Higher Homologues of Histamine on the Human Histamine H3 Receptor: Effect of Various Substitutions at the Primary Amino Function-Reference-Cited by-同舟云学术

A Chemical Switch for the Modulation of the Functional Activity of Higher Homologues of Histamine on the Human Histamine H3 Receptor: Effect of Various Substitutions at the Primary Amino Function

Published:2006-03-22 Issue:8 Volume:49 Page:2549-2557
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Govoni Marinella¹,Lim Herman D.¹,El-Atmioui Dris¹,Menge Wiro M. P. B.¹,Timmerman Henk¹,Bakker Remko A.¹,Leurs Rob¹,De Esch Iwan J. P.¹

Affiliation:

1. Leiden/Amsterdam Center for Drug Research, Department of Pharmacochemistry, Vrije Universiteit Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0504353

Reference74 articles.

1. Molecular pharmacological aspects of histamine receptors

2. Cloning and Functional Expression of the Human Histamine H3Receptor

3. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

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