Design, Synthesis, and Structure–Activity Relationships of Novel Pyrazolo[5,1-b]thiazole Derivatives as Potent and Orally Active Corticotropin-Releasing Factor 1 Receptor Antagonists-Reference-Cited by-同舟云学术

Design, Synthesis, and Structure–Activity Relationships of Novel Pyrazolo[5,1-b]thiazole Derivatives as Potent and Orally Active Corticotropin-Releasing Factor 1 Receptor Antagonists

Published:2012-10-01 Issue:19 Volume:55 Page:8450-8463
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Takahashi Yoshinori,Hashizume Minako,Shin Kogyoku,Terauchi Taro,Takeda Kunitoshi,Hibi Shigeki¹,Murata-Tai Kaoru,Fujisawa Masae,Shikata Kodo,Taguchi Ryota,Ino Mitsuhiro,Shibata Hisashi,Yonaga Masahiro

Affiliation:

1. Project Management, Head Office, Eisai Co., Ltd., 4-20-22 Koishikawa, Bunkyo-ku, Tokyo 112-8088, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300864p

Reference34 articles.

1. Characterization of a 41-Residue Ovine Hypothalamic Peptide That Stimulates Secretion of Corticotropin and β-Endorphin

2. Molecular Properties of the CRF Receptor

3. Expression cloning of a human corticotropin-releasing-factor receptor.

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