Design and Synthesis of Histidine Analogues of Folic Acid and Methotrexate as Potential Folylpolyglutamate Synthetase Inhibitors-Reference-Cited by-同舟云学术

Design and Synthesis of Histidine Analogues of Folic Acid and Methotrexate as Potential Folylpolyglutamate Synthetase Inhibitors

Published:1996-01-01 Issue:21 Volume:39 Page:4340-4344
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mao Zhenmin¹,Pan Jianping¹,Kalman Thomas I.¹

Affiliation:

1. Department of Medicinal Chemistry, School of Pharmacy, State University of New York at Buffalo, Buffalo, New York 14260

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960250j

Reference34 articles.

1. McGuire, J. J.; Coward, J. K. Pteroylpolyglutamates: Biosynthesis, Degradation, and Function. InFolates and Pterins,Vol.1; Blakley, R. L., Benkovic, S. J., Eds.; John Wiley & Sons: New York, 1984; pp 135−190.

2. Chromosomal assignment of the gene for folylpolyglutamate synthetase to human chromosome 9

3. The Biosynthesis of Folic Acid

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