Identification and Synthesis of a Novel Selective Partial PPARδ Agonist with Full Efficacy on Lipid Metabolism In Vitro and In Vivo-Reference-Cited by-同舟云学术

Identification and Synthesis of a Novel Selective Partial PPARδ Agonist with Full Efficacy on Lipid Metabolism In Vitro and In Vivo

Published:2007-03-08 Issue:7 Volume:50 Page:1495-1503
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sauerberg Per¹,Olsen Grith S.¹,Jeppesen Lone¹,Mogensen John P.¹,Pettersson Ingrid¹,Jeppesen Claus B.¹,Daugaard Jens R.¹,Galsgaard Elisabeth D.¹,Ynddal Lars¹,Fleckner Jan¹,Panajotova Vladimira¹,Polivka Zdenek¹,Pihera Pavel¹,Havranek Miroslav¹,Wulff Erik M.¹

Affiliation:

1. Novo Nordisk A/S, Diabetes Research Unit, Novo Nordisk Park, 2760 Måløv, Denmark, and RE&D VUFB, Podebradska 56/186, 180 66 Praha 9, Czech Republic

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm061202u

Reference34 articles.

1. Activation of a member of the steroid hormone receptor superfamily by peroxisome proliferators

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3. A systematic review of the clinical effectiveness of pioglitazone in the treatment of type 2 diabetes mellitus

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