Calpain 10 Homology Modeling with CYGAK and Increased Lipophilicity Leads to Greater Potency and Efficacy in Cells-Reference-Cited by-同舟云学术

Calpain 10 Homology Modeling with CYGAK and Increased Lipophilicity Leads to Greater Potency and Efficacy in Cells

Published:2012-05-31 Issue:8 Volume:7 Page:1410-1419
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Smith Matthew A.¹,McInnes Campbell²,Whitaker Ryan M.¹,Lindsey Christopher C.¹,Comer Richard F.¹,Beeson Craig C.¹,Schnellmann Rick G.¹³

Affiliation:

1. Center for Cell Death, Injury, and Regeneration, Department of Pharmaceutical and Biomedical Sciences, Medical University of South Carolina, Charleston, South Carolina 29425, United States

2. Department of Pharmaceutical and Biomedical Sciences, University of South Carolina, Columbia, South Carolina 29208, United States

3. Ralph Johnson VA Medical Center, Charleston, South Carolina 29401, United States

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cb300219h

Reference42 articles.

1. Inhibitors of calpain activation (PD150606 and E-64) and renal ischemia-reperfusion injury

2. The Calpain System

3. Structure, Activation, and Biology of Calpain

4. Calpain inhibitor-1 reduces renal ischemia/reperfusion injury in the rat

5. Calpain Inhibitor SNJ-1945 Attenuates Events Prior to Angiogenesis in Cultured Human Retinal Endothelial Cells

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