Convergent Asymmetric Synthesis of Two Complex TRPV1 Antagonists-Reference-Cited by-同舟云学术

Convergent Asymmetric Synthesis of Two Complex TRPV1 Antagonists

Published:2011-08-08 Issue:5 Volume:15 Page:1192-1200
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Butcher Kenneth J.¹,Denton Steven M.¹,Field Stuart E.¹,Gillmore Adam T.¹,Harbottle Gareth W.¹,Howard Roger M.¹,Laity Daniel A.¹,Ngono Christian J.¹,Pibworth Benjamin A.¹

Affiliation:

1. Pfizer Worldwide Research and Development, Sandwich Laboratories, Ramsgate Road, Sandwich CT13 9NJ, United Kingdom

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op200177b

Reference22 articles.

1. Analgesic potential of TRPV1 antagonists

2. Vanilloid Receptor TRPV1 Antagonists as the Next Generation of Painkillers. Are We Putting the Cart before the Horse?

3. The Discovery of Capsazepine, the First Competitive Antagonist of the Sensory Neuron Excitants Capsaicin and Resiniferatoxin

4. α-Substituted N-(4-tert-butylbenzyl)-N′-[4-(methylsulfonylamino)benzyl]thiourea analogues as potent and stereospecific TRPV1 antagonists

5. Hester, J B.U.S. Patent 5,155,268 A, 1992.

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