α-Substituted β-Oxa Isosteres of Fosmidomycin: Synthesis and Biological Evaluation-Reference-Cited by-同舟云学术

α-Substituted β-Oxa Isosteres of Fosmidomycin: Synthesis and Biological Evaluation

Published:2012-07-11 Issue:14 Volume:55 Page:6566-6575
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Brücher Karin¹,Illarionov Boris²,Held Jana³,Tschan Serena³,Kunfermann Andrea⁴,Pein Miriam K.¹,Bacher Adelbert⁴,Gräwert Tobias²,Maes Louis⁵,Mordmüller Benjamin³⁶,Fischer Markus²,Kurz Thomas¹

Affiliation:

1. Institut für Pharmazeutische und Medizinische Chemie, Heinrich Heine Universität, Universitätsstr. 1, 40225 Düsseldorf, Germany

2. Hamburg School of Food Science, Universität Hamburg, Grindelallee 117, 20146 Hamburg, Germany

3. Institut für Tropenmedizin, Eberhard Karls Universität Tübingen, Wilhelmstr. 27, 72074 Tübingen, Germany

4. Center for Integrated Protein Science Munich, Lehrstuhl für Biochemie, Technische Universität München, Lichtenbergstr. 4, 85747 Garching, Germany

5. Laboratory for Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Groenenborgerlaan 171, 2020 Wilrijk, Belgium

6. Medical Research Unit, Albert Schweitzer Hospital, Lambaréné, Gabon

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300652f

Reference57 articles.

1. Malarial Parasites vs. Antimalarials: Never-Ending Rumble in the Jungle

2. Evidence of Artemisinin-Resistant Malaria in Western Cambodia

3. Emergence of artemisinin-resistant malaria on the western border of Thailand: a longitudinal study

4. New medicines to improve control and contribute to the eradication of malaria

Cited by 35 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. 1-Deoxy-d-xylulose 5-phosphate reductoisomerase as target for anti Toxoplasma gondii agents: crystal structure, biochemical characterization and biological evaluation of inhibitors;Biochemical Journal;2024-08-21

2. Reverse N-Substituted Hydroxamic Acid Derivatives of Fosmidomycin Target a Previously Unknown Subpocket of 1-Deoxy-d-xylulose 5-Phosphate Reductoisomerase (DXR);ACS Infectious Diseases;2024-04-22

3. Inhibition of DXR in the MEP pathway with lipophilic N-alkoxyaryl FR900098 analogs;RSC Medicinal Chemistry;2024

4. Design and synthesis of fosmidomycin analogs containing aza‐linkers and their biological activity evaluation;Pest Management Science;2023-10-17

5. Synthesis of bis-α-hydroxyphosphine oxides based on salicyl aldehyde scaffold;Журнал общей химии;2023-01-15