Identification of Bacteria-Selective Threonyl-tRNA Synthetase Substrate Inhibitors by Structure-Based Design-Reference-Cited by-同舟云学术

Identification of Bacteria-Selective Threonyl-tRNA Synthetase Substrate Inhibitors by Structure-Based Design

Published:2013-02-12 Issue:4 Volume:56 Page:1748-1760
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Teng Min¹,Hilgers Mark T.¹,Cunningham Mark L.¹,Borchardt Allen¹,Locke Jeffrey B.¹,Abraham Sunny¹,Haley Gregory¹,Kwan Bryan P.¹,Hall Courtney¹,Hough Grayson W.¹,Shaw Karen J.¹,Finn John¹

Affiliation:

1. Medicinal Chemistry, ‡Structural Biology, §Biology, and ∥Analytical Chemistry, Trius Therapeutics, Inc., 6310 Nancy Ridge Drive, San Diego, California 92121, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301756m

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