Design and Synthesis of a Novel Photoaffinity Ligand for the Dopamine and Serotonin Transporters Based on 2β-Carbomethoxy-3β-biphenyltropane-Reference-Cited by-同舟云学术

Design and Synthesis of a Novel Photoaffinity Ligand for the Dopamine and Serotonin Transporters Based on 2β-Carbomethoxy-3β-biphenyltropane

Published:2006-10-05 Issue:22 Volume:49 Page:6621-6625
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Newman Amy Hauck¹,Cha Joo Hwan¹,Cao Jianjing¹,Kopajtic Theresa¹,Katz Jonathan L.¹,Parnas M. Laura¹,Vaughan Roxanne¹,Lever John R.¹

Affiliation:

1. Medicinal Chemistry and Psychobiology Sections, National Institute on Drug AbuseIntramural Research Program, National Institutes of Health, Department of Health and Human Services, Baltimore, Maryland, University of North Dakota School of Medicine, Grand Forks, North Dakota, University of MissouriColumbia, Departments of Radiology and Medical Pharmacology and Physiology, and Harry S. Truman Veterans Administration Medical Center, Columbia, Missouri

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0603973

Reference21 articles.

1. Probes for the dopamine transporter: New leads toward a cocaine-abuse therapeutic?A focus on analogues of benztropine and rimcazole

2. Recognition of Benztropine by the Dopamine Transporter (DAT) Differs from That of the Classical Dopamine Uptake Inhibitors Cocaine, Methylphenidate, and Mazindol as a Function of a DAT Transmembrane 1 Aspartic Acid Residue

3. A novel photoaffinity label for the dopamine transporter based on N-substituted 3α-[bis(4′-fluorophenyl)methoxy]tropane

4. Dopamine Transporter Ligand Binding Domains

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