Evolution of a Compact Photoprobe for the Dopamine Transporter Based on (±)-threo-Methylphenidate-Reference-Cited by-同舟云学术

Evolution of a Compact Photoprobe for the Dopamine Transporter Based on (±)-threo-Methylphenidate

Published:2012-03-20 Issue:5 Volume:3 Page:378-382
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Lapinsky David J.¹,Yarravarapu Nageswari¹,Nolan Tammy L.¹,Surratt Christopher K.¹,Lever John R.²³,Tomlinson Michael⁴,Vaughan Roxanne A.⁴,Deutsch Howard M.⁵

Affiliation:

1. Division of Pharmaceutical Sciences, Duquesne University, 600 Forbes Avenue, Pittsburgh, Pennsylvania 15282, United States

2. Departments of Radiology, and Medical Pharmacology and Physiology, One Hospital Drive, University of Missouri, Columbia, Missouri 65212, United States

3. Harry S. Truman Veterans Administration Medical Center, 800 Hospital Drive, Columbia, Missouri 65201, United States

4. Department of Biochemistry and Molecular Biology, University of North Dakota School of Medicine and Health Sciences, Grand Forks, North Dakota 58202, United States

5. School of Chemistry and Biochemistry, Georgia Institute of Technology, Atlanta, Georgia 30332, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml3000098

Reference30 articles.

1. Recognition of Benztropine by the Dopamine Transporter (DAT) Differs from That of the Classical Dopamine Uptake Inhibitors Cocaine, Methylphenidate, and Mazindol as a Function of a DAT Transmembrane 1 Aspartic Acid Residue

2. A novel photoaffinity ligand for the dopamine transporter based on pyrovalerone

3. Azido-iodo-N-benzyl derivatives of threo-methylphenidate (Ritalin, Concerta): Rational design, synthesis, pharmacological evaluation, and dopamine transporter photoaffinity labeling

4. (±)-2-(N-tert-Butylamino)-3′-[125I]-iodo-4′-azidopropiophenone: A dopamine transporter and nicotinic acetylcholine receptor photoaffinity ligand based on bupropion (Wellbutrin, Zyban)

5. Relationship between Conformational Changes in the Dopamine Transporter and Cocaine-Like Subjective Effects of Uptake Inhibitors

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