Synthesis and Benzodiazepine Receptor Affinity of Pyrazolo[1,5-a]pyrimidine Derivatives. 3. New 6-(3-Thienyl) Series as α1 Selective Ligands-Reference-Cited by-同舟云学术

Synthesis and Benzodiazepine Receptor Affinity of Pyrazolo[1,5-a]pyrimidine Derivatives. 3. New 6-(3-Thienyl) Series as α1 Selective Ligands

Published:2002-12-11 Issue:2 Volume:46 Page:310-313
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Selleri Silvia¹,Bruni Fabrizio¹,Costagli Camilla¹,Costanzo Annarella¹,Guerrini Gabriella¹,Ciciani Giovanna¹,Gratteri Paola¹,Bonaccini Claudia¹,Malmberg Aiello Petra¹,Besnard François¹,Renard Stephane¹,Costa Barbara¹,Martini Claudia¹

Affiliation:

1. Department of Pharmaceutical Sciences, University of Firenze, Via G. Capponi 9, 50121 Firenze, Italy, Department of Preclinical and Clinical Pharmacology, University of Firenze, Viale Pieraccini 6, 50139 Firenze, Italy, Department of Molecular and Functional Genomics, Synthélabo, 10 Rue des Carrîeres, 92500 Rueil-Malmaison, France, and Departments of Psychiatry, Neurobiology, Pharmacology, and Biotechnologies, University of Pisa, Via Bonanno 6, 56126 Pisa, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020999w

Reference15 articles.

1. Synthesis and BZR affinity of pyrazolo[1,5- a ]pyrimidine derivatives. part 1: study of the structural features for BZR recognition

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