Preparation and Evaluation at the Delta Opioid Receptor of a Series of Linear Leu-Enkephalin Analogues Obtained by Systematic Replacement of the Amides-Reference-Cited by-同舟云学术

Preparation and Evaluation at the Delta Opioid Receptor of a Series of Linear Leu-Enkephalin Analogues Obtained by Systematic Replacement of the Amides

Published:2013-05-20 Issue:8 Volume:4 Page:1204-1216
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Rochon Kristina¹,Proteau-Gagné Arnaud¹,Bourassa Philippe¹,Nadon Jean-François¹,Côté Jérome¹,Bournival Véronique¹,Gobeil Fernand¹,Guérin Brigitte¹,Dory Yves L.¹,Gendron Louis¹

Affiliation:

1. Département de Physiologie et Biophysique, ‡Laboratoire de Synthèse Supramoléculaire, Département de Chimie, §Département de pharmacologie, and ∥Département de Médecine Nucléaire et Radiobiologie, Institut de Pharmacologie, Université de Sherbrooke, 3001, 12e Avenue Nord, Sherbrooke, Québec J1H 5N4, Canada

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/cn4000583

Reference74 articles.

1. Endogenous opiates and behavior: 2011

2. Opioids: first lessons from knockout mice

3. Differential noxious and motor tolerance of chronic delta opioid receptor agonists in rodents

4. A Comparison of the Antinociceptive and Adverse Effects of the mu-Opioid Agonist Morphine and the delta-Opioid Agonist SNC80

5. The role of δ-opioid receptor subtypes in neuropathic pain

Cited by 22 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. The impact of multifunctional enkephalin analogs and morphine on the protein changes in crude membrane fractions isolated from the rat brain cortex and hippocampus;Peptides;2024-04

2. Stapling of leu-enkephalin analogs with bifunctional reagents for prolonged analgesic activity;Chemical Communications;2024

3. Modification and Delivery of Enkephalins for Pain Modulation;International Journal of Pharmaceutics;2023-11

4. Amide-to-ester substitution as a stable alternative to N-methylation for increasing membrane permeability in cyclic peptides;Nature Communications;2023-03-17

5. Peptidomimetics and Their Applications for Opioid Peptide Drug Discovery;Biomolecules;2022-09-05