New Histamine H3-Receptor Ligands of the Proxifan Series: Imoproxifan and Other Selective Antagonists with High Oral in Vivo Potency-Reference-Cited by-同舟云学术

New Histamine H3-Receptor Ligands of the Proxifan Series: Imoproxifan and Other Selective Antagonists with High Oral in Vivo Potency

Published:2000-08-01 Issue:17 Volume:43 Page:3335-3343
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sasse Astrid¹,Sadek Bassem¹,Ligneau Xavier¹,Elz Sigurd¹,Pertz Heinz H.¹,Luger Peter¹,Ganellin C. Robin¹,Arrang Jean-Michel¹,Schwartz Jean-Charles¹,Schunack Walter¹,Stark Holger¹

Affiliation:

1. Institut für Pharmazie, Freie Universität Berlin, Königin-Luise-Strasse 2+4, 14195 Berlin, Germany; Laboratoire Bioprojet, 30 rue des Francs-Bourgeois, 75003 Paris, France; Institut für Chemie/Kristallographie, Freie Universität Berlin, Takustrasse 6, 14195 Berlin, Germany; Department of Chemistry, Christopher Ingold Laboratories, University College London, 20 Gordon Street, London WC1H 0AJ, U.K.; and Unité de Neurobiologie et Pharmacologie Moléculaire (U. 109), Centre Paul Broca de l'INSERM, 2ter rue...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm000971p

Reference47 articles.

1. Stark, H.; Elz, S.; Ligneau, X.; Sadek, B.; Krause, M.; Pertz, H.; Arrang, J.M.; Ganellin, C. R.; Schwartz, J.C.; Schunack, W. Proxifans, a Novel Series of Histamine H3-Receptor Antagonists with High Selectivity and High Oral in Vivo CNS Potency. 37th IUPAC Congress and 27th GDCh General Meeting, Berlin, Germany, Aug 14−19, 1999; Abstract-CD-ROM 287, APP-1-014.

2. Three loci related to the src oncogene and tyrosine-specific protein kinase activity in Drosophila

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